Buspirone

Anxiolytic (non-benzodiazepine, 5-HT1A)
Drug Class
Anxiolytic (non-benzodiazepine, 5-HT1A)
Mechanism of Action (MOA)
Partial agonist at serotonin 5-HT1A receptors.
Clinical Notes
Generalized anxiety — not a controlled substance; label reports no abuse potential, tolerance or dependence, and lacks prominent sedation.
Source
FDA label

Sources

Reviewed September 2026
  1. FDA label — FDA / DailyMed

Checked against the guideline or standard reference the exam keys to. If it has moved, use Report an error below.

Used for

Same family

Anxiolytics, sedatives & hypnotics · 3 drugs

Got a pharmacology lecture that covers Buspirone? Turn it into flashcards and board-style questions, free. Drop it on the home page

All pharmacology